Ganellin, C. R., and Stanley M. Roberts. Medicinal Chemistry: The Role of Organic Chemistry in Drug Research. 2nd ed. London: Academic Press, 1993.
King, Frank D. and Royal Society of Chemistry (Great Britain). Medicinal Chemistry: Principles and Practice. 2nd ed. Cambridge: Royal Society of Chemistry, 2002.
Patrick, Graham L. An Introduction to Medicinal Chemistry. Seventh edition. Oxford: Oxford University Press, 2023.
Strømgaard, Kristian, Povl Krogsgaard-Larsen, and Ulf Madsen. Textbook of Drug Design and Discovery. 5th ed. Boca Raton: CRC Press, 2017. https://ebookcentral.proquest.com/lib/nottingham/detail.action?docID=4617075.
Wermuth, C. G. The Practice of Medicinal Chemistry. 4th ed. London: Elsevier Academic Press, 2015. http://www.sciencedirect.com/science/book/9780124172050.