Ganellin, C. R., and Stanley M. Roberts. Medicinal Chemistry: The Role of Organic Chemistry in Drug Research. 2nd ed, Academic Press, 1993.
King, Frank D. and Royal Society of Chemistry (Great Britain). Medicinal Chemistry: Principles and Practice. 2nd ed, Royal Society of Chemistry, 2002.
Patrick, Graham L. An Introduction to Medicinal Chemistry. Seventh edition, Oxford University Press, 2023.
Strømgaard, Kristian, et al. Textbook of Drug Design and Discovery. 5th ed, CRC Press, 2017, https://ebookcentral.proquest.com/lib/nottingham/detail.action?docID=4617075. Electronic resource.
Wermuth, C. G. The Practice of Medicinal Chemistry. 4th ed, Elsevier Academic Press, 2015, http://www.sciencedirect.com/science/book/9780124172050. Electronic resource.