Ganellin CR and Roberts SM, Medicinal Chemistry: The Role of Organic Chemistry in Drug Research (2nd ed, Academic Press 1993)
King FD and Royal Society of Chemistry (Great Britain), Medicinal Chemistry: Principles and Practice (2nd ed, Royal Society of Chemistry 2002)
Patrick GL, An Introduction to Medicinal Chemistry (Seventh edition, Oxford University Press 2023)
Strømgaard K, Krogsgaard-Larsen P and Madsen U, Textbook of Drug Design and Discovery (5th ed, CRC Press 2017) <https://ebookcentral.proquest.com/lib/nottingham/detail.action?docID=4617075>
Wermuth CG, The Practice of Medicinal Chemistry (4th ed, Elsevier Academic Press 2015) <http://www.sciencedirect.com/science/book/9780124172050>